Find out how to combat elevated estradiol on PCT with the aromatase inhibitor Exemestane, what dosages to use and how long to take. No other member of the aromatase inhibitor class has these properties. Using exemestane in bodybuilding after a course of steroids, an athlete can not only quickly restore the processes of testosterone synthesis, but due to an increase in the concentration of insulin-like growth factor, it shifts the balance between anabolism and catabolism towards the former.
Some builders are confident that this has a positive effect on the recovery of the body, because the rollback effect is minimized and muscle tissue is protected from destruction. However, if you understand the immediate results of using exemestane in bodybuilding after a course of steroids, it becomes clear that this is undesirable. Summing up the conversation about the positive effects of the drug, we will highlight the most significant:
- An excellent means of preventing gynecomastia.
- Effectively suppresses the level of female hormones.
- Promotes anabolic growth.
- Improves muscle definition.
- It is a good means of preventing hypertension.
- Reduces the negative effect of estrogen on the work of the pituitary arch.
How Exemestane works
When the drug is used for medical purposes, it deprives cancer cells of the estrogen necessary for their vital activity. There is no doubt about the effectiveness of using aromazine for these purposes. However, it is recommended to use tamoxifen first. If this drug does not give positive results, it is worth starting to use exemestane.
However, even with high efficiency, this drug is used in medicine less often than anastrozole. This is due to the fact that arimidex behaves in many ways similar to the primary aromatase inhibitor. Moreover, this happens not only in the treatment of breast cancer after menopause, but also during the treatment of other oncological ailments.
However, we are more interested in the mechanisms of exemestane in relation to the suppression of the negative effects of anabolic steroids. Having become acquainted with the properties and effects of the drug, it is already possible to draw certain conclusions in this matter. It is important to remember that estrogen-type side effects may not appear when using steroids.
If we talk specifically about estrogenic side effects, then for their development, the AAS used by the athlete must have the ability to aromatize or progestogenic activity. The primary aromatizing anabolic is testosterone. However, drugs based on substances derived from this hormone can enhance the work of estrogens. Methandienone is a prime example of this.
Also, boldenone can be attributed to such steroids, the ability of which to aromatize is 50 percent of the dough. This is not enough for a rapid increase in the concentration of female hormones. Among the steroids that can cause estrogenic side effects are trenbolone and nandrolone. They are weakly aromatized, but at the same time they have strong progestogenic activity.
This may be enough for female hormone levels to rise above normal limits. This largely depends on the genetic characteristics of the organism. Trenbolone is not able to interact with the aromatase enzyme, however, due to the high progestogenic activity, the development of gynecomastia is possible. This happens again, with the genetic predisposition of the athlete. If these drugs are used in conjunction with aromatizing AAS, the risks of developing estrogen-type side effects increase.
Regardless of the anabolic used, exemestane can protect you from side effects. In sports, steroids are actively used, which are based on substances derived from dihydrotestosterone. In principle, they are not capable of aromatizing. An exception to this rule is oxymetholone, which has estrogenic activity. However, it is not able to aromatize and aromazine will not be effective on the course of Anapolon.
Now let's look at the mechanisms of the aromatase inhibitor, which are manifested when using exemestane in bodybuilding after a course of steroids. You should know that on an anabolic cycle, the synthesis of endogenous male hormone is suppressed. The extent of this negative effect of AAS depends on the steroids used and their dosage. However, even the lightest drug can negatively affect the work of the pituitary axis.
After the end of the anabolic cycle, the body will begin to synthesize testosterone again, but only after all exogenous hormones have been utilized. This will take a long time frame. Much depends on the characteristics of the athlete's body and in the worst case can take about a year. It is quite obvious that such a situation is unacceptable. PCT is carried out precisely with the aim of accelerating the secretion of endogenous male hormone.
In itself, the state of low dough is abnormal, but additional negative aspects appear. In particular, levels of muscle-damaging cortisol increase and libido decreases. We have already noted that aromazine is able to accelerate the synthesis of testosterone.
In this case, the drug is characterized by a low androgenic activity, and it accelerates the secretion of insulin-like growth factor. All this leads to the fact that some athletes start using exemestane in bodybuilding after a course of steroids. At the same time, they forget about the main purpose of this drug - inhibition of the aromatase enzyme.
There is no doubt that a high concentration of estrogen leads to undesirable consequences for a man. But the balance between female and male hormones is also extremely important. Scientists have proven that estradiol regulates the balance of lipoprotein compounds, normalizes the body's defense mechanisms and affects libido. The main task of restorative therapy after anabolic cycles is to stimulate the processes of testosterone secretion. But at the same time, it is important to remember about the normalization of the work of all body systems. If the level of estrogen is strongly suppressed, then this is simply impossible to achieve. This is why we do not recommend using exemestane in bodybuilding after a steroid cycle. The drug can be most useful during an anabolic cycle, but not after its completion.
Instructions for the use of Exemestane in bodybuilding
The recommended dosages of the drug are in the range of 12.5 to 25 milligrams, and it must be consumed every second day. However, in most cases, athletes should only use 12.5 milligrams of exemestane no more than three times a week.
If the maximum allowed dose is used, then the duration of such a course of exemestane should not be long. It is worth using 25 milligrams only if the cholesterol balance is disturbed, and in other situations, limit yourself to the minimum dosage. Also in professional sports, exemestane is sometimes used one or two weeks before the start of a tournament to improve muscle definition.